(2-Morpholin-4-yl-4-phenyl-1,3-thiazol-5-yl)methanol Chemical Properties,Usage,Production
Uses
Androgen receptor-IN-3 (Compound 22) is an androgen receptor inhibitor. Androgen receptor-IN-3 inhibits AR-driven transcriptional activity in LNCaP cells, with an IC50 of 5.04 μM[1].
References
[1] Li H, et al. Discovery of small-molecule inhibitors selectively targeting the DNA-binding domain of the human androgen receptor. J Med Chem. 2014 Aug 14;57(15):6458-67. DOI:10.1021/jm500802j
