ChemicalBook CAS数据库列表 CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
- CAS号:115044-69-4
- 英文名:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
- 中文名:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
- CBNumber:CB7217236
- 分子式:C103H185N31O24S
- 分子量:2273.83
- MOL File:115044-69-4.mol
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)化学性质
- 密度 :1.37±0.1 g/cm3(Predicted)
- 储存条件 :−20°C
- 溶解度 :Soluble in DMSO
- 形态 :White lyophilized solid
- 颜色 :white
- 水溶解性 :water: soluble
安全信息
- 安全说明 :22-24/25
- WGK Germany :3
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)性质、用途与生产工艺
- 生物活性 Calmodulin-Dependent Protein Kinase II (290-309) 是有效的 CaMK 拮抗剂, 抑制抑制Ca2+/钙调蛋白依赖性蛋白激酶II的 IC50 值为52 nM。
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靶点
IC50: 52 nM (calmodulin-dependent protein kinase II)
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体外研究
Peptide 290 to 309 is found to be a potent calmodulin antagonist with an IC 50 of 52 nM for inhibition of Ca 2+ /calmodulin-dependent protein kinase. Neither truncation from the amino terminus (peptide 296-309) nor extension in the carboxyl-terminal direction (peptide 294-319) markedly affects calmodulin binding, whereas shortening the peptide from the carboxyl terminus (peptide 290-302) or from both ends (peptide 295-304) results in the elimination of this activity.
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)上下游产品信息
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下游产品
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) 试剂级价格
- 更新日期:2023/03/20
- 产品编号:HY-P1479
- 产品名称:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) Calmodulin-Dependent Protein Kinase II (290-309)
- CAS编号:115044-69-4
- 包装:1 mg
- 价格:3300元
- 更新日期:2023/03/20
- 产品编号:HY-P1479
- 产品名称:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) Calmodulin-Dependent Protein Kinase II (290-309)
- CAS编号:115044-69-4
- 包装:5mg
- 价格:13000元
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)生产厂家
- 公司名称:Carbosynth
- 联系电话:--
- 电子邮件:sales@carbosynth.com
- 国家:英国
- 产品数:6005
- 优势度:58
- 公司名称:VWR
- 联系电话:--
- 电子邮件:solutions@vwr.com
- 国家:英国
- 产品数:6548
- 优势度:82