生物活性 靶点 体外研究 CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) 试剂级价格
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CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)

CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309),115044-69-4,结构式
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
  • CAS号:115044-69-4
  • 英文名:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
  • 中文名:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)
  • CBNumber:CB7217236
  • 分子式:C103H185N31O24S
  • 分子量:2273.83
  • MOL File:115044-69-4.mol
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)化学性质
  • 密度 :1.37±0.1 g/cm3(Predicted)
  • 储存条件 :−20°C
  • 溶解度 :Soluble in DMSO
  • 形态 :White lyophilized solid
  • 颜色 :white
  • 水溶解性 :water: soluble
安全信息

CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)性质、用途与生产工艺

  • 生物活性 Calmodulin-Dependent Protein Kinase II (290-309) 是有效的 CaMK 拮抗剂, 抑制抑制Ca2+/钙调蛋白依赖性蛋白激酶II的 IC50 值为52 nM。
  • 靶点

    IC50: 52 nM (calmodulin-dependent protein kinase II)

  • 体外研究

    Peptide 290 to 309 is found to be a potent calmodulin antagonist with an IC 50 of 52 nM for inhibition of Ca 2+ /calmodulin-dependent protein kinase. Neither truncation from the amino terminus (peptide 296-309) nor extension in the carboxyl-terminal direction (peptide 294-319) markedly affects calmodulin binding, whereas shortening the peptide from the carboxyl terminus (peptide 290-302) or from both ends (peptide 295-304) results in the elimination of this activity.

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CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) 试剂级价格
  • 更新日期:2023/03/20
  • 产品编号:HY-P1479
  • 产品名称:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) Calmodulin-Dependent Protein Kinase II (290-309)
  • CAS编号:115044-69-4
  • 包装:1 mg
  • 价格:3300元
  • 更新日期:2023/03/20
  • 产品编号:HY-P1479
  • 产品名称:CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309) Calmodulin-Dependent Protein Kinase II (290-309)
  • CAS编号:115044-69-4
  • 包装:5mg
  • 价格:13000元
CALMODULIN-DEPENDENT PROTEIN KINASE II (290-309)生产厂家
  • 公司名称:Service Chemical Inc.
  • 联系电话:--
  • 电子邮件:sales@chemos-group.com
  • 国家:德国
  • 产品数:6350
  • 优势度:71