ChemicalBook CAS数据库列表 DerMorphin Trifluoroacetate
DerMorphin Trifluoroacetate
- CAS号:78331-26-7
- 英文名:DerMorphin Trifluoroacetate
- 中文名:DerMorphin Trifluoroacetate
- CBNumber:CB32652493
- 分子式:C42H51F3N8O12
- 分子量:916.91
- MOL File:78331-26-7.mol
DerMorphin Trifluoroacetate化学性质
- 熔点 :157-162°C
- 储存条件 :-20°C Freezer
- 溶解度 :DMSO (Slightly), Methanol (Slightly)
- 形态 :Solid
- 颜色 :White
DerMorphin Trifluoroacetate性质、用途与生产工艺
- 生物活性 Dermorphin TFA 是在两栖类皮肤中发现的一种天然七肽 μ-阿片受体 (MOR) 激动剂。Dermorphin 可用于抑制神经痛。
-
靶点
μ-opioid receptor (MOR)
-
体外研究
Dermorphin, a peptide isolated from the skin of Phyllomedusa frogs and the peptide receptor (NOP) component by the endogenous agonist nociceptin/orphanin FQ (N/OFQ). In displacement binding studies at CHO hMu , Dermorphin and DeNo displac the binding of [ 3 H]-DPN in a concentration dependent and saturable manner. Dermorphin displays an affinity of 7.17, while N/OFQ fails to displace [ 3 H]-DPN at the Delta receptor. Dermorphin and DeNo stimulate the binding of GTPγ[ 35 S] in a concentration dependent and saturable manner at the Mu receptor.
DerMorphin Trifluoroacetate上下游产品信息
上游原料
下游产品
DerMorphin Trifluoroacetate生产厂家
- 公司名称：TargetMol Chemicals Inc.
- 联系电话：+1-781-999-5354
- 电子邮件：support@targetmol.com
- 国家：美国
- 产品数：19973
- 优势度：58
- 公司名称：MedChemExpress
- 联系电话：--
- 电子邮件：sales@medchemexpress.com
- 国家：美国
- 产品数：6398
- 优势度：58
