BB-Cl-Amidine hydrochloride
- CAS号:
- 英文名:BB-Cl-Amidine hydrochloride
- 中文名:BB-Cl-Amidine hydrochloride
- CBNumber:CB05419683
- 分子式:C??H??Cl?N?O
- 分子量:0
- MOL File:Mol file
BB-Cl-Amidine hydrochloride性质、用途与生产工艺
- 生物活性 BB-Cl-Amidine hydrochloride 是肽基精氨酸脱胺酶 (PAD) 的抑制剂。
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靶点
PAD.
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体内研究
Treatment with BB-Cl-amidine subtly reduces splenomegaly in MRL/lpr mice, while there is a trend towards increased circulating levels of anti-NET antibodies with PAD inhibitor treatment. However, neither PAD inhibitor affected body weight or total IgG levels. Indeed, treatment with both Cl-amidine and BB-Cl-amidine significantly improves endothelium-dependent vasorelaxation. The BB-Cl-amidine group also shows a strong trend towards downregulation of IRGs. Treatment with either Cl-amidine or BB-Cl-amidine significantly improves muzzle alopecia, in many cases preventing it entirely.
Animal Model: MRL/lpr mice. Dosage: 1 mg/kg. Administration: Subcutaneous injection daily from 8 to 14 weeks of age. Result: Significantly improved endothelium-dependent vasorelaxation and showed a strong trend towards downregulation of IRGs.
BB-Cl-Amidine hydrochloride上下游产品信息
上游原料
下游产品
BB-Cl-Amidine hydrochloride 试剂级价格- 更新日期:2024/08/19
- 产品编号:HY-111347A
- 产品名称:BB-Cl-Amidine hydrochloride BB-Cl-Amidine hydrochloride
- CAS编号:
- 包装:1mg
- 价格:450元
- 更新日期:2024/08/19
- 产品编号:HY-111347A
- 产品名称:BB-Cl-Amidine hydrochloride BB-Cl-Amidine hydrochloride
- CAS编号:
- 包装:5mg
- 价格:950元
BB-Cl-Amidine hydrochloride生产厂家
- 公司名称:天津普西唐生物医药科技有限公司
- 联系电话:010-60605840 15801484223;
- 电子邮件:psaitong@jm-bio.com
- 国家:中国
- 产品数:29778
- 优势度:58