103614-28-4
中文名称
化合物 T23963
英文名称
dynorphin A ethylamide (1-9), MeTyr(1)-MeArg(7)-Leu(8)-
CAS
103614-28-4
分子式
C56H93N19O10
分子量
1192.46
MOL 文件
103614-28-4.mol
结构式
基本信息
中文别名
化合物 T23963
英文别名
Daeatal
dynorphin A ethylamide (1-9), MeTyr(1)-MeArg(7)-Leu(8)-
L-Argininamide, N-methyl-L-tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-L-arginyl-N2-methyl-L-arginyl-D-leucyl-N-ethyl- (9CI)
dynorphin A ethylamide (1-9), MeTyr(1)-MeArg(7)-Leu(8)-
L-Argininamide, N-methyl-L-tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-L-arginyl-N2-methyl-L-arginyl-D-leucyl-N-ethyl- (9CI)
应用领域
用途一
Dynorphin A ethylamide (1-9), The opioid activities were examined in the bioassays (guinea pig ileum, mouse vas deferens and rabbit vas deferens). the extension of the C-terminal in the peptide chain of [MeArg7,D-Leu8]-Dyn(1-8)-NH2 analogues by Arg is ineffective for increasing the kappa-opioid activities, kappa-receptor selectivity and/or analgesic effects of the peptides.