67121-76-0

Fluperlapine is an agonist of the serotonin 5-HT6/5-HT7 receptors.

ChEBI: Fluperlapine is a benzazepine.

Seven metabolites of fluperlapine are detected by culturing with incubation of human hepatocytes. The major metabolite is the N-oxide and the formation of sulfates remains high although decreases with time in the culture. Two glucuronides found in vivo are not detected in any of the cultures.