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Piperidylthiambutene is a potent μ-opioid receptor (MOR) agonist with a Ki of 2.75 nM. Piperidylthiambutene exhibits analgesic and antitussive properties and can be utilized in relevant research[1].

[1] De Luca MA, et al. Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists. Neuropharmacology. 2022 Dec 15;221:109263. DOI:10.1016/j.neuropharm.2022.109263