264622-53-9

MRS1706 is a selective adenosine A_2B receptor inverse agonist with K_i values of 1.39, 157, 112, and 230 nM for human A_2B, A₁, A_2A, and A₃ receptors, respectively.

MRS 1706 is a selective and potent Adenosine A2B-R inverse agonist Ki (binding affinity) values of 1.39, 157, 112, and 230 nM for human A2B, A1, A2A, and A3 receptors, respectively.

Potent and selective adenosine A 2B receptor inverse agonist (K i values are 1.39, 157, 112 and 230 nM for human A 2B , A 1 , A 2A and A 3 receptors respectively).