2470126-25-9

Sitagliptin N-sulfate is a phase II metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor (–)-sitagliptin (Item No. 13252).1 Sitagliptin N-sulfate is formed via sulfation and has been found in rat bile following oral administration of (–)-sitagliptin.WARNING This product is not for human or veterinary use.

[1] MARIA G BECONI. Disposition of the dipeptidyl peptidase 4 inhibitor sitagliptin in rats and dogs.[J]. Drug Metabolism and Disposition, 2007, 35 4: 525-532. DOI: 10.1124/dmd.106.013110