170964-68-8

Name	8-cyclohexyl-2,3,3a,4,5,6-hexahydro-1H-pyrazino[3,2,1-jk]carbazole methanesulfonate
CAS	170964-68-8
Molecular Formula	C21H30N2O3S
Molecular Weight	390.54
MOL File	170964-68-8.mol

Synonyms

8-cyclohexyl-2,3,3a,4,5,6-hexahydro-1H-pyrazino[3,2,1-jk]carbazole methanesulfonate

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Chemical Properties

solubility	Soluble to 100 mM in DMSO
form	Powder
color	White to off-white

Hazard Information

Uses

Tetrindole Mesylate is part of a pharmaceutical composition, which exhibits anti-cancer effects for preventing and treating prostate cancer.

Definition

ChEBI:Tetrindole mesylate is a racemate composed of equimolar amounts of (R)- and (S)-tetrindole mesylate. It has a role as an antidepressant, an EC 1.4.3.4 (monoamine oxidase) inhibitor and a serotonergic agonist. It contains a (R)-tetrindole mesylate and a (S)-tetrindole mesylate.

in vivo

Tetrindole mesylate (25 mg/kg; po; single dose) inhibits rat brain and liver mitochondrial MAO A by 80% within 0.5-1 hr and the onset of recovery of enzyme activity became evident after 24 hr in male albino rats weighing 180-200 g^[1].

IC 50

MAO-A

Spectrum Detail

8-cyclohexyl-2,3,3a,4,5,6-hexahydro-1H-pyrazino[3,2,1-jk]carbazole methanesulfonate(170964-68-8)¹HNMR

Supplier

MedBioPharmaceutical Technology Inc

Telephone021-69568360 18916172912

Websitehttp://www.med-bio.cn/

Shanghai Yifei Biotechnology Co. , Ltd.

Telephone021-65675885 18964387627

Websitehttp://www.efebio.com

Nanjing Shizhou Biology Technology Co.,Ltd

Telephone025-85560043 15850508050

Websitehttp://www.synzest.com

TargetMol Chemicals Inc.

Telephone 15002134094

Websitehttps://www.targetmol.cn/

Shanghai Amole Biotechnology Co., Ltd.

Telephone13370042665 18916960931

Websitehttps://www.amole.com.cn/

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