153049-49-1

Name	PD 145065
CAS	153049-49-1
Molecular Formula	C52H67N7O10
MDL Number	MFCD00467202
Molecular Weight	950.13
MOL File	153049-49-1.mol

Synonyms

PD 145065 Ac-bhg-Leu-Asp-Ile-Ile-Trp AC-DBHG-LEU-ASP-ILE-ILE-TRP AC-D-BHG-LEU-ASP-ILE-ILE-TRP-OH [AC-DBHG16] ENDOTHELIN-1 (16-21) endothelin receptor antagonist*pd 145065 N-Acetyl-α-[10,11-Dihydro-5H-dibenzo[a,d]cycloheptadien-5-yl]-D-Gly-Leu-Asp-Ile-Ile-Trp L-Tryptophan, N-[N-[N-[N-[N-[N-acetyl-D-2-(10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)glycyl]-L-leucyl]-L-α-aspartyl]-L-isoleucyl]-L-isoleucyl]- (9CI)

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Chemical Properties

storage temp.	−20°C
solubility	phosphate buffer, pH 7.5: 1mg/mL
form	White solid
color	white

Safety Data

WGK Germany

Hazard Information

Biological Activity

Cell permeable: no''Primary Target
Endothelin receptor antagonist''Product does not compete with ATP.''Reversible: no''Target IC50: 4 nM against endothelin receptor (ETA receptor) in rabbit renal artery vascular smooth muscle cells; 15 nM for the ETB receptor (r at cerebellum)

Supplier

GL Biochem (Shanghai) Ltd

Telephone21-61263452 13641803416

Websitehttp://www.glschina.com/

Nanjing Peptide Biotech Ltd.

Telephone025-025-58361106-805-805 13082558573

Websitehttp://www.njpeptide.com

Hangzhou Peptidego Biotech Co.,Ltd.

Telephone0571-87213919

Websitehttp://www.peptidego.com

Nanjing Meihao Pharmaceutical Technology Co., Ltd.

Telephonemeitaochem@126.com

Websitehttps://www.chemicalbook.com/ShowSupplierProductsList31244/0.htm

Hangzhou Sinoda Pharmaceutical Technology Co. LTD

Telephone0571-87213919 17306812703

Websitehttps://www.chemicalbook.com/ShowSupplierProductsList1355681/0.htm

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