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LY2228820
- русский язык имя
- английское имяLY2228820
- CAS №862507-23-1
- CBNumberCB82518277
- ФормулаC26H37FN6O6S2
- мольный вес612.7369832
- номер MDLMFCD22572532
- файл Mol862507-23-1.mol
химическое свойство
температура хранения | Store at -20°C |
растворимость | ≥30.65 mg/mL in DMSO; ≥45 mg/mL in H2O with ultrasonic; ≥9.9 mg/mL in EtOH with ultrasonic |
форма | solid |
цвет | White to yellow |
FDA UNII | QUW7B71FO9 |
LY2228820 химические свойства, назначение, производство
Использование
LY2228820 is a novel and potent p38MAPK inhibitor with potent antiinflammatory activity. LY2228820 significantly inhibited phosphorylation of MAPKAPK2 and/or HSP27, down stream targets of p38MAPK, in both multiple myeloma (MM) cell lines and LT-BMSCs. LY2228820 is a potential candidate to improve MM patient outcome both by enhancing the effect of Bortezomib (B675700) and by reducing osteoskeletal events.LY2228820 поставщик
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