ADRA1D receptor agonist 1
英文名称:ADRA1D receptor agonist 1
CAS号:1191908-14-1
分子式:C15H14Cl2N4O
分子量:337.2
EINECS号:
Mol文件:1191908-14-1.mol
ADRA1D receptor agonist 1 用途与合成方法
ADRA1D receptor agonist 1 (compound (R)-9S) 是一个高效、选择性的,有口服活性的 α1D 肾上腺素受拮抗剂,Ki 值为 1.6 nM。
Ki: 1.6 nM (α 1D adrenoceptor)
ADRA1D receptor agonist 1 shows low hERG inhibition.
ADRA1D receptor agonist 1 exhibits higher selectivity for α1D-AR over α1A- and α1B-ARs .
ADRA1D receptor agonist 1 (4.4 µg/kg; i.v.) dose-dependently decreases the non-voiding bladder contractions during the urinary storage phase in rats with BOO.
Animal Model: | Rat with bladder outlet obstruction (BOO) |
Dosage: | 4.4 µg/kg |
Administration: | Intravenous injection |
Result: | Dose-dependently decreased the non-voiding bladder contractions during urinary storage phase in rats with BOO. |
ADRA1D receptor agonist 1 价格(试剂级)
更新日期 | 产品编号 | 产品名称 | CAS号 | 包装 | 价格 |
---|---|---|---|---|---|
2024-11-08 | HY-135270 | 1 mg | 2181 | ||
2024-11-08 | HY-135270 | 5 mg | 4800 |
ADRA1D receptor agonist 1供应商 更多
天津普西唐生物医药科技有限公司
联系电话:010-60605840 15801484223;
产品介绍:
英文名称:ADRA1D receptor agonist 1
CAS:1191908-14-1
包装信息:100mg
备注: 试剂级
上海一飞生物科技有限公司
联系电话:021-65675885 18964387627
产品介绍:
英文名称:ADRA1D receptor agonist 1
CAS:1191908-14-1
纯度:98%
包装信息:2mg;25mg;50mg
备注:试剂级
TargetMol中国(陶术生物)
联系电话: 15002134094
产品介绍:
中文名称:ADRA1D receptor antagonist 1 盐酸盐
英文名称:ADRA1D receptor antagonist 1 HCl
CAS:1191908-14-1
纯度:98.13%
包装信息:1mg/RMB 1780