Paliperidone

• Product Name:Paliperidone
• Synonyms: Paliperidone (Invega) 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-Methyl- Risperidone EP IMpurity C Paliperidone 9-Hydroxyrisperidone 9-Hydroxyrisperidone solution Racemic Paliperidone 4h-pyrido(2,1-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluro-1,2-benzis oxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-
• CAS:144598-75-4
• MF:C23H27FN4O3
• MW:426.48
• EINECS:620-493-1
• Mol File:144598-75-4.mol
• 

Paliperidone, (±)-3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one(Invega), is essentially insoluble in water and is available asextended-release tablets. Paliperidone is delivered at a constantrate using an osmotic drug release device (OsmoticRelease Oral Systems [OROS]). The absolute bioavailabilityof paliperidone is 28%, and studies in healthy subjects on ahigh-fat, high-calorie meal showed an increase in AUC.Paliperidone is 74% bound to plasma proteins. After a single,1-mg dose of C-paliperidone, 59% of the dose was excretedin the urine as unchanged drug, and 32% of the dose was recoveredas metabolites. Most of the drug (80%) is excreted bythe kidneys. Paliperidone is metabolized by dealkylation, hydroxylation,dehydrogenation, and scission of the benzoxazolering. None of these metabolic pathways account for morethan 10% of the dose. The terminal elimination half-life ofpaliperidone is 23 hours.

• Paliperidone
• 
• US $0.00-0.00/Kg/Bag
• CAS:144598-75-4
• Min. Order: 1Kg/Bag
• Purity: 0.99
• Supply Ability: 20 tons
• 2024-11-21

• Paliperidone
• 
• US $0.00 /g
• CAS:144598-75-4
• Min. Order: 1g
• Purity: More Than 99%
• Supply Ability: 100kg/Month
• 2024-11-18

• Company Name:Zhuzhou focus pharmaceutical technology co., LTD
• Tel: +86-13776644403
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:98% Package:1g;5g;10g;25g;50g;100g;bulk More...
• CB Index:58
• Related Information:Catalog(1984)

• Company Name:Shandong Risen-Sun Pharmaceutical Co., Ltd
• Tel:+8615621883869 15621883869
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:99% HPLC Package:5KG;1KG
• CB Index:58
• Related Information:Catalog(108)

• Company Name:NanJing Vtrying Pharmatech Co.,Ltd
• Tel: 17314186806
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:99.5% HPLC Package:10g;100g;1kg;5kg;25kg
• CB Index:58
• Related Information:Catalog(86)

• Company Name:Hefei Lifeon Pharmaceutical Co.Ltd.
• Tel:0551-65328450 18956095011
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:99% Package:1KG;5KG
• CB Index:58
• Related Information:Catalog(23)

• Company Name:J & K SCIENTIFIC LTD.
• Tel:010-82848833 400-666-7788
• Products Intro:Product Name:Paliperidone, 99%, a potent D2 and 5-HT2A antagonist
  CAS:144598-75-4
  Purity:99% Package:10MG;50MG More...
• CB Index:76
• Related Information:Catalog(94657)

• Company Name:Chemvon Biotechnology Co., Ltd
• Tel:021-50790412
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:99% HPLC Package:1g;50g;100g;1kg More...
• CB Index:57
• Related Information:Catalog(371)

• Company Name:Meryer (Shanghai) Chemical Technology Co., Ltd.
• Tel:021-61259108 18621169109
• Products Intro:Product Name:Paliperidone
  CAS:144598-75-4
  Purity:>97.0%(T) Package:200Mg;1g Remarks:P1897 More...
• CB Index:62
• Related Information:Catalog(40228)