FAK/Aurora kinase-IN-1 is a FAK and aurora kinase inhibitor with IC50 values of 6.61 nM and 0.91 nM, respectively. FAK/Aurora kinase-IN-1 shows anticancer effects (WO2018019252A1; compound 11)[1].
References
[1] Wenlai Zhou, et al. Novel fused pyridine derivatives useful as fak/aurora kinase inhibitors. WO2018019252A1.