1403947-26-1

LAS191954 is a potent, selective and orally active PI3Kδ inhibitor for inflammatory diseases treatment, with an IC50 of 2.6 nM[1].

PI3Kδ: 2.6 nM (IC₅₀)

Store at -20°C

[1] Erra M, et al. Discovery of a Potent, Selective, and Orally Available PI3Kδ Inhibitor for the Treatment of Inflammatory Diseases. ACS Med Chem Lett. 2016 Nov 30;8(1):118-123. DOI:10.1021/acsmedchemlett.6b00438