118101-09-0

L-365,260 is a non-peptide competitive CCK-BR antagonist.

ChEBI: L-365260 is a benzodiazepine.

Selective cholecystokinin receptor 2 (CCK 2 ) antagonist (IC 50 values are 2 and 280 nM at CCK 2 and CCK 1 receptors respectively) that is inactive at a range of other receptors including opiate, muscarinic acetylcholine, α - and β adrenergic, histamine, angiotensin and bradykinin receptors.

Store at +4°C