ChemicalBook CAS数据库列表 AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
- CAS号:167114-91-2
- 英文名:AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
- 中文名:AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE
- CBNumber:CB7671283
- 分子式:C64H116N22O19
- 分子量:1497.74
- MOL File:167114-91-2.mol
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE化学性质
- 储存条件 :-20°C
- 溶解度 :H2O: soluble
- 形态 :lyophilized powder
- 颜色 :white
- 水溶解性 :Soluble to 1 mg/ml in water
安全信息
- 危险品标志 :Xn,F
- 危险类别码 :20/21/22-36-11
- 安全说明 :22-24/25-26-36/37-16
- WGK Germany :3
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE性质、用途与生产工艺
- 生物活性 Autocamtide-2-related inhibitory peptide 是高度特异性的、CaMKII 的有效抑制剂,其IC50 值为 40 nM。
-
靶点
IC50: 40 nM (CaMKII).
-
体外研究
It is found that Autocamtide-2-related inhibitory peptide (a novel synthetic peptide ATP) is a potent inhibitor of CaM-kinase II with an IC 50 of 40 nM, which is active in the presence or absence of Ca 2+ /calmodulin. It is 50 and 500 times more potent than CaMK-(281-302Ala286) and KN-93,respectively, under the assay condition used.
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE上下游产品信息
上游原料
下游产品
AUTOCAMTIDE-2-RELATED INHIBITORY PEPTIDE生产厂家
- 公司名称:Carbosynth
- 联系电话:--
- 电子邮件:sales@carbosynth.com
- 国家:英国
- 产品数:6018
- 优势度:58
- 公司名称:TOCRIS-US
- 联系电话:--
- 电子邮件:customerservice@tocris.co.uk
- 国家:英国
- 产品数:5729
- 优势度:77
- 公司名称:VWR
- 联系电话:--
- 电子邮件:solutions@vwr.com
- 国家:英国
- 产品数:6554
- 优势度:82
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